Found 5 Enz. Inhib. hit(s) with Target = 'Protein mono-ADP-ribosyltransferase PARP10' and Ligand = 'BDBM50446130'
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
Health & Science University
Curated by ChEMBL
Health & Science University
Curated by ChEMBL
Affinity DataIC50: 562nMAssay Description:Inhibition of full length recombinant human His6-tagged PARP10 expressed in Escherichia coli BL21(DE3) preincubated for 15 mins followed by biotinyla...More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
Health & Science University
Curated by ChEMBL
Health & Science University
Curated by ChEMBL
Affinity DataIC50: 562nMAssay Description:Inhibition of full length recombinant human His6-tagged PARP10 expressed in Escherichia coli BL21(DE3) preincubated for 15 mins followed by biotinyla...More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
Health & Science University
Curated by ChEMBL
Health & Science University
Curated by ChEMBL
Affinity DataIC50: 570nMAssay Description:Inhibition of full length recombinant human His6-tagged PARP10 expressed in Escherichia coli BL21(DE3) preincubated for 15 mins followed by biotinyla...More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
Health & Science University
Curated by ChEMBL
Health & Science University
Curated by ChEMBL
Affinity DataIC50: 2.31E+3nMAssay Description:Inhibition of recombinant human His6-tagged PARP10 ADP-ribosyltransferase domain expressed in Escherichia coli BL21(DE3) preincubated for 15 mins fol...More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
Health & Science University
Curated by ChEMBL
Health & Science University
Curated by ChEMBL
Affinity DataKd: 3.10E+3nMAssay Description:Binding affinity to PARP10 (unknown origin) assessed as apparent dissociation constantMore data for this Ligand-Target Pair