Found 2 Enz. Inhib. hit(s) with Target = 'Protein mono-ADP-ribosyltransferase PARP14' and Ligand = 'BDBM50397961'
TargetProtein mono-ADP-ribosyltransferase PARP14(Homo sapiens (Human))
Karolinska Institutet
Curated by ChEMBL
Karolinska Institutet
Curated by ChEMBL
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of hexahistidine-tagged human recombinant ARTD8 catalytic domain (1611 to 1801 amino acids) expressed in Escherichia coli BL21(DE3) assess...More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Homo sapiens (Human))
Karolinska Institutet
Curated by ChEMBL
Karolinska Institutet
Curated by ChEMBL
Affinity DataKd: 1.12E+4nMAssay Description:Binding affinity at human recombinant ARTD8 expressed in Escherichia coli BL21 (DE3) R3 pRARE cells by isothermal titration calorimetryMore data for this Ligand-Target Pair