Found 2 Enz. Inhib. hit(s) with Target = 'Protein mono-ADP-ribosyltransferase PARP3' and Ligand = 'BDBM50250875'
TargetProtein mono-ADP-ribosyltransferase PARP3(Homo sapiens (Human))
University Of Oslo
Curated by ChEMBL
University Of Oslo
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ARTD3 (unknown origin) measured after 4 hrs in presence of NAD+ by fluorescence assayMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP3(Homo sapiens (Human))
University Of Oslo
Curated by ChEMBL
University Of Oslo
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human PARP3 using NAD+ as substrate by fluorescence assayMore data for this Ligand-Target Pair