Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Protein-arginine deiminase type-4' and Ligand = 'BDBM52947'
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM52947((2Z,4S,4aR,5S,5aR,6R,12aS)-2-[amino(hydroxy)methyl...)
Affinity DataKi:  6.30E+5nMAssay Description:Inhibition of PAD4 measured by intercept plot of Lineweaver-Burke analysesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM52947((2Z,4S,4aR,5S,5aR,6R,12aS)-2-[amino(hydroxy)methyl...)
Affinity DataIC50:  8.60E+5nMAssay Description:Inhibition of PAD4 by ABPP-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed