Found 2 Enz. Inhib. hit(s) with Target = 'Protein-glutamine gamma-glutamyltransferase 2' and Ligand = 'BDBM50241218'
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
University Of Ottawa
Curated by ChEMBL
University Of Ottawa
Curated by ChEMBL
Affinity DataKi: 3.80E+3nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
University Of Ottawa
Curated by ChEMBL
University Of Ottawa
Curated by ChEMBL
Affinity DataKi: 1.29E+4nMAssay Description:Irreversible inhibition of human TG2 using AL5 as substrate by colorimetric assayMore data for this Ligand-Target Pair