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Found 2 Enz. Inhib. hit(s) with Target = 'Proteinase-activated receptor 1' and Ligand = 'BDBM50031414'
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50031414(1-{(S)-2-[(S)-2-((S)-2-{(S)-2-[(S)-2-((S)-2-Amino-...)
Affinity DataEC50:  3.00E+3nMAssay Description:Activation of PAR-1 in human platelet-rich plasma assessed as induction of platelet aggregation by turbidimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50031414(1-{(S)-2-[(S)-2-((S)-2-{(S)-2-[(S)-2-((S)-2-Amino-...)
Affinity DataEC50:  500nMAssay Description:Evaluated for the activation of human thrombin receptor measured by platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed