Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'Proteinase-activated receptor 1' and Ligand = 'BDBM50031432'
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50031432((S)-2-{(S)-2-[(S)-2-((S)-2-Amino-propionylamino)-3...)
Affinity DataEC50:  130nMAssay Description:Evaluated for the activation of human thrombin receptor measured by platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed