Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'Proteinase-activated receptor 1' and Ligand = 'BDBM50179584'
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50179584((+)-(3R,3aS,4S,4aR,8aS,9aR)-3-methyl-4-(2-(6-(3-(t...)
Affinity DataIC50:  300nMAssay Description:Displacement of [3H]haTRAP from PAR1 in human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed