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Found 3 Enz. Inhib. hit(s) with Target = 'Pyroglutamylated RF-amide peptide receptor' and Ligand = 'BDBM50347819'
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50347819(CHEMBL1802414 | P550)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]-43RFa from human QRFP receptor expressed in CHO cells by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50347819(CHEMBL1802414 | P550)
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50347819(CHEMBL1802414 | P550)
Affinity DataEC50:  4.90nMAssay Description:Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed