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Found 2 Enz. Inhib. hit(s) with Target = 'Pyruvate kinase' and Ligand = 'BDBM50192869'
TargetPyruvate kinase(Staphylococcus aureus (strain MRSA252))
Simon Fraser University

Curated by ChEMBL
LigandPNGBDBM50192869(CIS-3,4-DIHYDROHAMACANTHIN B)
Affinity DataIC50:  16nMAssay Description:Inhibition of recombinant N-terminal His-tagged methicillin-resistant Staphylococcus aureus MRSA252 pyruvate kinase expressed in Escherichia coli BL2...More data for this Ligand-Target Pair
TargetPyruvate kinase(Staphylococcus aureus (strain MRSA252))
Simon Fraser University

Curated by ChEMBL
LigandPNGBDBM50192869(CIS-3,4-DIHYDROHAMACANTHIN B)
Affinity DataIC50:  16nMAssay Description:Inhibition of methicillin-resistant Staphylococcus aureus pyruvate kinase by coupled lactate dehydrogenase continuous assayMore data for this Ligand-Target Pair