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Found 1 Enz. Inhib. hit(s) with Target = 'Pyruvate kinase PKM' and Ligand = 'BDBM114395'
TargetPyruvate kinase PKM(Homo sapiens (Human))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM114395(7,11b-dihydro-6H-indeno[2,1-c][1]benzopyran-3,4,6a...)
Affinity DataIC50:  3.40E+5nMAssay Description:Inhibition of PKM2 (unknown origin) Ser362, Lys367, Lys207, Ser77, Asp177, Asp178, Asn75, Gly52, Gly128 residuesMore data for this Ligand-Target Pair
In DepthDetails PubMed