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Found 4 Enz. Inhib. hit(s) with Target = 'RAC-beta serine/threonine-protein kinase' and Ligand = 'BDBM50373459'
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50373459(CHEMBL258696)
Affinity DataIC50:  212nMAssay Description:Inhibition of Akt2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50373459(CHEMBL258696)
Affinity DataIC50:  212nMAssay Description:Inhibition of Akt2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50373459(CHEMBL258696)
Affinity DataIC50:  276nMAssay Description:Inhibition of Akt2 by cell-based IPKA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50373459(CHEMBL258696)
Affinity DataIC50:  730nMAssay Description:Inhibition of Akt2 by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed