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Found 3 Enz. Inhib. hit(s) with Target = 'RAC-gamma serine/threonine-protein kinase' and Ligand = 'BDBM15148'
TargetRAC-gamma serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM15148(2,3-diphenylquinoxaline 1 | 2-[4-(3-phenylquinoxal...)
Affinity DataIC50: >5.00E+4nMAssay Description:Purified recombinant human Akt1, Akt2, and Akt3 proteins were monitored for kinase activity in the presence or absence of Akt inhibitors in a 96-well...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-gamma serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM15148(2,3-diphenylquinoxaline 1 | 2-[4-(3-phenylquinoxal...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human recombinant Akt3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-gamma serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM15148(2,3-diphenylquinoxaline 1 | 2-[4-(3-phenylquinoxal...)
Affinity DataIC50: >2.50E+5nMAssay Description:Inhibition of Akt3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed