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Found 2 Enz. Inhib. hit(s) with Target = 'RAC-gamma serine/threonine-protein kinase' and Ligand = 'BDBM15162'
TargetRAC-gamma serine/threonine-protein kinase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM15162(2-(4-{[4-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-y...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Akt3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-gamma serine/threonine-protein kinase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM15162(2-(4-{[4-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-y...)
Affinity DataIC50: >5.00E+4nMAssay Description:Purified recombinant human Akt1, Akt2, and Akt3 proteins were monitored for kinase activity in the presence or absence of Akt inhibitors in a 96-well...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed