Found 5 Enz. Inhib. hit(s) with Target = 'Receptor-interacting serine/threonine-protein kinase 2' and Ligand = 'BDBM13336'
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
University Of Iowa
Curated by ChEMBL
University Of Iowa
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of human receptor-interacting serine-threonine kinase 2 (RIPK2) at 100 uM ATPMore data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
University Of Iowa
Curated by ChEMBL
University Of Iowa
Curated by ChEMBL
Affinity DataKd: 2.10E+3nMAssay Description:Average Binding Constant for RIPK2; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
University Of Iowa
Curated by ChEMBL
University Of Iowa
Curated by ChEMBL
Affinity DataKd: 24nMAssay Description:Binding constant for RIPK2 kinase domainMore data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
University Of Iowa
Curated by ChEMBL
University Of Iowa
Curated by ChEMBL
Affinity DataKd: 24nMAssay Description:Binding constant for RIPK2 kinase domainMore data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
University Of Iowa
Curated by ChEMBL
University Of Iowa
Curated by ChEMBL
Affinity DataKd: 24nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair