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Found 3 Enz. Inhib. hit(s) with Target = 'Regulator of G-protein signaling 16' and Ligand = 'BDBM47798'
TargetRegulator of G-protein signaling 16(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM47798(4-chloranyl-6-(4,6-dimethylpyrimidin-2-yl)sulfanyl...)
Affinity DataKi:  4.21E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 16(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM47798(4-chloranyl-6-(4,6-dimethylpyrimidin-2-yl)sulfanyl...)
Affinity DataEC50:  1.63E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 16(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM47798(4-chloranyl-6-(4,6-dimethylpyrimidin-2-yl)sulfanyl...)
Affinity DataEC50:  5.19E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay