Found 7 Enz. Inhib. hit(s) with Target = 'Retinoic acid receptor RXR-gamma' and Ligand = 'BDBM50032667'
Affinity DataKi: 299nMAssay Description:Binding affinity towards recombinantly expressed Retinoic acid receptor RXR-gamma in baculoviral sysytem, by using 5 nM [3H]-targretin in a competiti...More data for this Ligand-Target Pair
Affinity DataEC50: 246nMAssay Description:Ability to activate gene expression at Retinoic acid receptor RXR-gamma was evaluated in a cotransfection assay.More data for this Ligand-Target Pair
Affinity DataKd: 299nMAssay Description:Binding affinity to Retinoic acid receptor RXR-gamma was evaluated in a competitive binding assay.More data for this Ligand-Target Pair
Affinity DataKd: 424nMAssay Description:Inhibition of [3H]-9-cis-RA binding to baculovirus expressed retinoid receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 246nMAssay Description:Transcriptional activity was evaluated in CV-1 cells transfected with expression vector for Retinoic acid receptor RXR-gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 246nMAssay Description:Effective concentration against retinoid receptor isoform (RXR gamma) expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20E+3nMAssay Description:Effective concentrations against Retinoic acid receptor RXR-gammaMore data for this Ligand-Target Pair