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Found 4 Enz. Inhib. hit(s) with Target = 'Sentrin-specific protease 1' and Ligand = 'BDBM50421700'
TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM50421700(CHEMBL5289965)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human recombinant His6 tagged SENP1 catalytic domain expressed in Escherichia coli BL21 (DE3) using SUMO1-AMC as substrate incubated fo...More data for this Ligand-Target Pair
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TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM50421700(CHEMBL5289965)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of human recombinant His6 tagged SENP1 catalytic domain expressed in Escherichia coli BL21 (DE3) using SUMO3-AMC as substrate incubated fo...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM50421700(CHEMBL5289965)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of human recombinant His6 tagged SENP1 catalytic domain expressed in Escherichia coli BL21 (DE3) using SUMO2-AMC as substrate incubated fo...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM50421700(CHEMBL5289965)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human recombinant SENP1 catalytic domain expressed in Escherichia coli BL21 (DE3) using SUMO1-AMC as substrate incubated for 10 mins fo...More data for this Ligand-Target Pair
In DepthDetails PubMed