Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase 17B' and Ligand = 'BDBM50559222'
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))
University Of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50559222(CHEMBL4752776)
Affinity DataIC50:  34nMAssay Description:Inhibition of human STK17B in presence of ATP at Km levelMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))
University Of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50559222(CHEMBL4752776)
Affinity DataIC50:  34nMAssay Description:Inhibition of N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli incubated for 90 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))
University Of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50559222(CHEMBL4752776)
Affinity DataIC50:  190nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))
University Of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50559222(CHEMBL4752776)
Affinity DataKd:  5.60nMAssay Description:Binding affinity to human STK17B assessed as displacement of immobilized ligand by KINOMEscan scanMAX assay relative to controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))
University Of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50559222(CHEMBL4752776)
Affinity DataKd:  5.60nMAssay Description:Binding affinity to N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli by KINOMEscan scan...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB