Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase B-raf' and Ligand = 'BDBM50176328'
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50176328((3-(2-phenyl-5-(pyridin-4-yl)-1H-imidazol-4-yl)phe...)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibition bRaf kinase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50176328((3-(2-phenyl-5-(pyridin-4-yl)-1H-imidazol-4-yl)phe...)
Affinity DataKd: >196nMAssay Description:Binding affinity at bRaf kinase in fluorescent ligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed