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Found 2 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase B-raf' and Ligand = 'BDBM50176334'
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50176334(5-(2-(1-amino-2-methylpropan-2-yl)-5-(pyridin-4-yl...)
Affinity DataIC50:  6nMAssay Description:Inhibition bRaf kinase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50176334(5-(2-(1-amino-2-methylpropan-2-yl)-5-(pyridin-4-yl...)
Affinity DataKd:  4.80nMAssay Description:Binding affinity at bRaf kinase in fluorescent ligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed