Found 4 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase BRSK2' and Ligand = 'BDBM2579'
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Inhibition of human BRSK2 using KKLNRTLSFAEPG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataIC50: 3.30nMAssay Description:Inhibition of human BRSK2 using KKLNRTLSFAEPG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataKd: 3.5nMAssay Description:Binding constant for BRSK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataKd: 3.5nMAssay Description:Binding constant for full-length BRSK2More data for this Ligand-Target Pair