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Found 2 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase Chk1' and Ligand = 'BDBM50375267'
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375267(CHEMBL410195)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of recombinant Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375267(CHEMBL410195)
Affinity DataEC50:  70nMAssay Description:Inhibition of human Chk1 in H1299 cells assessed as blockade of Cdc25A degradationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed