Found 3 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase Chk2' and Ligand = 'BDBM4814'
Affinity DataIC50: 17nMAssay Description:Inhibition of CHK2 using biotinylated substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence microplate ...More data for this Ligand-Target Pair
Affinity DataKd: 7.10nMAssay Description:Binding affinity to CHEK2More data for this Ligand-Target Pair
Affinity DataKd: 10nMAssay Description:Binding constant for CHEK2 kinase domainMore data for this Ligand-Target Pair