Found 4 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase D3' and Ligand = 'BDBM2579'
TargetSerine/threonine-protein kinase D3(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human PKCnu using KKLNRTLSVA as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase D3(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataIC50: 2.10nMAssay Description:Inhibition of human PKCnu using KKLNRTLSVA as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase D3(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataKd: 18nMAssay Description:Binding constant for PRKD3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase D3(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataKd: 18nMAssay Description:Binding constant for PRKD3 kinase domainMore data for this Ligand-Target Pair