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Found 1 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase MARK2' and Ligand = 'BDBM247038'
TargetSerine/threonine-protein kinase MARK2(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM247038(2-((1R,3aR, 6S,7R,7aS)-5,5- difluoro-7- ((E)-2-(5-...)
Affinity DataIC50:  2.62nMAssay Description:This assay measures the potency of the inventive compounds as PAR-1 receptor antagonists.Frozen HEK 293 Cells were plated in 384-well PDL coated plat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent