Found 2 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase PAK 1' and Ligand = 'BDBM50097134' TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Inhibition of human recombinant PAK1 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate assessed as substrate phosphorylation...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Shanghai Chempartner
Curated by ChEMBL
Shanghai Chempartner
Curated by ChEMBL
Affinity DataIC50: 281nMAssay Description:Inhibition of PAK1 in human EBC1 cells assessed as inhibition of MEK phosphorylation at S298 after 2 hrs by HTRF assayMore data for this Ligand-Target Pair
