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Found 2 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase PLK1' and Ligand = 'BDBM50297961'
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297961(3-(2-chlorobenzyloxy)-5-(imidazo[1,2-a]pyridin-3-y...)
Affinity DataIC50:  35nMAssay Description:Inhibition of PLK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50297961(3-(2-chlorobenzyloxy)-5-(imidazo[1,2-a]pyridin-3-y...)
Affinity DataEC50:  1.15E+3nMAssay Description:Inhibition of PLK1-mediated mitosis in human HeLaS3 cells after 18 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed