Found 8 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase PLK2' and Ligand = 'BDBM2579'
Affinity DataKi: 150nMAssay Description:Kinase was assayed in 384-well polypropylene plate format. The compound was mixed with kinase and biotinylated peptide substrate and incubated. After...More data for this Ligand-Target Pair
Affinity DataIC50: 328nMAssay Description:Inhibition of human PLK2 using casein as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 366nMAssay Description:Inhibition of PLK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 471nMAssay Description:Inhibition of human PLK2 using casein as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 957nMAssay Description:Inhibition human recombinant full length GST-tagged Plk2 expressed in baculovirus expression system after 1 hr by FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
Affinity DataIC50: 957nMAssay Description:Inhibition of recombinant full length human GST-tagged PLK2 expressed in baculovirus expression system using ser/thr 16 as substrate incubated for 1 ...More data for this Ligand-Target Pair
Affinity DataKd: 200nMAssay Description:Binding constant for PLK2 kinase domainMore data for this Ligand-Target Pair