Found 4 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase ULK1' and Ligand = 'BDBM50271371'
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))
Sichuan Universitt China Hospital
Curated by ChEMBL
Sichuan Universitt China Hospital
Curated by ChEMBL
Affinity DataEC50: 19nMAssay Description:Activation of recombinant human N-terminal GST-tagged ULK1 (1 to 649 residues) expressed in baculovirus infected Sf9 cells using MBP as substrate aft...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))
Sichuan Universitt China Hospital
Curated by ChEMBL
Sichuan Universitt China Hospital
Curated by ChEMBL
Affinity DataEC50: 19nMAssay Description:Antagonist potency against histamine H3 receptor in an electrically stimulated guinea pig ileumMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))
Sichuan Universitt China Hospital
Curated by ChEMBL
Sichuan Universitt China Hospital
Curated by ChEMBL
Affinity DataKd: 290nMAssay Description:Binding affinity to wild type ULK1 (unknown origin) expressed in HEK293T cells assessed as dissociation constant measured after 8 mins by SPR analysi...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))
Sichuan Universitt China Hospital
Curated by ChEMBL
Sichuan Universitt China Hospital
Curated by ChEMBL
Affinity DataEC50: 19nMAssay Description:Inhibition of ULK1 (unknown origin) using MBP as substrate after 60 mins by ADP-Glo assayMore data for this Ligand-Target Pair