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Found 4 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase ULK1' and Ligand = 'BDBM50271371'
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))
Sichuan Universitt China Hospital

Curated by ChEMBL
LigandPNGBDBM50271371(CHEMBL4125718)
Affinity DataEC50:  19nMAssay Description:Activation of recombinant human N-terminal GST-tagged ULK1 (1 to 649 residues) expressed in baculovirus infected Sf9 cells using MBP as substrate aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))
Sichuan Universitt China Hospital

Curated by ChEMBL
LigandPNGBDBM50271371(CHEMBL4125718)
Affinity DataEC50:  19nMAssay Description:Antagonist potency against histamine H3 receptor in an electrically stimulated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))
Sichuan Universitt China Hospital

Curated by ChEMBL
LigandPNGBDBM50271371(CHEMBL4125718)
Affinity DataKd:  290nMAssay Description:Binding affinity to wild type ULK1 (unknown origin) expressed in HEK293T cells assessed as dissociation constant measured after 8 mins by SPR analysi...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))
Sichuan Universitt China Hospital

Curated by ChEMBL
LigandPNGBDBM50271371(CHEMBL4125718)
Affinity DataEC50:  19nMAssay Description:Inhibition of ULK1 (unknown origin) using MBP as substrate after 60 mins by ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed