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Found 2 Enz. Inhib. hit(s) with Target = 'Serine protease 1' and Ligand = 'BDBM16309'
TargetSerine protease 1(Homo sapiens (Human))
Arris

LigandPNGBDBM16309(2-(quinolin-8-yl)-1H-1,3-benzodiazole-6-carboximid...)
Affinity DataKi:  8.04E+3nM ΔG°:  -28.8kJ/molepH: 8.2 T: 2°CAssay Description:Enzymes were incubated with inhibitors at eight inhibitor concentrations bracketing the Ki, prepared by serial dilution along with control lacking th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Arris

LigandPNGBDBM16309(2-(quinolin-8-yl)-1H-1,3-benzodiazole-6-carboximid...)
Affinity DataKi:  4.18E+4nMAssay Description:Enzymes were incubated with inhibitors at eight inhibitor concentrations bracketing the Ki, prepared by serial dilution along with control lacking th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed