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Found 2 Enz. Inhib. hit(s) with Target = 'Sigma non-opioid intracellular receptor 1' and Ligand = 'BDBM50082621'
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50082621((2S,6S,11S)-3-Benzyl-11-ethyl-1,2,3,4,5,6-hexahydr...)
Affinity DataKi:  26.7nMAssay Description:Affinity against Sigma opioid receptor type 1 using [3H]-(+)-Pentazocine in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50082621((2S,6S,11S)-3-Benzyl-11-ethyl-1,2,3,4,5,6-hexahydr...)
Affinity DataKi:  478nMAssay Description:Affinity against Sigma opioid receptor type 2 using [3H]- DTG in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed