Found 7 Enz. Inhib. hit(s) with Target = 'Sigma non-opioid intracellular receptor 1' and Ligand = 'BDBM94507'
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Medical College of Georgia
Curated by PDSP Ki Database
Medical College of Georgia
Curated by PDSP Ki Database
TargetSigma non-opioid intracellular receptor 1(RAT)
National Institute On Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute On Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Tested for its binding affinity towards sigma-1 site in presence of [3H]- dextromethorphanMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
National Institute On Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute On Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Tested for its binding affinity towards sigma-1 site in presence of [3H]- -(+)3 PPPMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Medical College of Georgia
Curated by PDSP Ki Database
Medical College of Georgia
Curated by PDSP Ki Database
Affinity DataKi: 19.5nMAssay Description:Binding affinity against Sigma receptor type 1 was determined by the displacement of [3H]pentazocine radioligandMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
National Institute On Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute On Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Tested for its binding affinity towards sigma-1 site in presence of [3H]- - (+) pentazocineMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
National Institute On Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute On Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 41nMAssay Description:Tested for its binding affinity towards sigma-1 site in rat brain using E3H1-(+)-SKF 10047 as radioligand in rat brainMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Medical College of Georgia
Curated by PDSP Ki Database
Medical College of Georgia
Curated by PDSP Ki Database
Affinity DataKi: 129nMAssay Description:Binding affinity to sigma-1 receptor (unknown origin)More data for this Ligand-Target Pair