Found 5 Enz. Inhib. hit(s) with Target = 'Small conductance calcium-activated potassium channel protein 1/2/3' and Ligand = 'BDBM50199404'
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 1.30E+3nMAssay Description:Displacement of [125I]apamin from SK channel in Wistar rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 1.30E+3nMAssay Description:Displacement of [125I]apamin from Wistar rat cortical apamin-sensitive siteMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 1.60E+3nMAssay Description:Inhibition of [125I]apamin binding to calcium-activated potassium (SK) channel of rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataIC50: 8.70E+3nMAssay Description:Inhibition of [125I]apamin binding to calcium-activated potassium (SK) channel of rat cortexMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataIC50: 1.50E+4nMAssay Description:Blockade of SK channel in Wistar rat brain assessed as inhibition of apamin-sensitive after-hyperpolarisationMore data for this Ligand-Target Pair