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Found 2 Enz. Inhib. hit(s) with Target = 'Sodium channel protein type 1 subunit alpha' and Ligand = 'BDBM492965'
TargetSodium channel protein type 1 subunit alpha(Homo sapiens (Human))
Xenon Pharmaceuticals

US Patent
LigandPNGBDBM492965(5-((2-bromo-3,6-difluorobenzyl)amino)-3-fluoro-6-m...)
Affinity DataIC50:  245nMAssay Description:This sodium influx assay employs the use of the cell permeable, sodium sensitive dye ANG2 to quantify sodium ion influx through sodium channels which...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium channel protein type 1 subunit alpha(Homo sapiens (Human))
Xenon Pharmaceuticals

US Patent
LigandPNGBDBM492965(5-((2-bromo-3,6-difluorobenzyl)amino)-3-fluoro-6-m...)
Affinity DataIC50:  245nMAssay Description:This sodium influx assay employs the use of the cell permeable, sodium sensitive dye ANG2 to quantify sodium ion influx through sodium channels which...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent