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Found 3 Enz. Inhib. hit(s) with Target = 'Sodium-dependent dopamine transporter' and Ligand = 'BDBM50453909'
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50453909(CHEMBL3084880)
Affinity DataKi:  78nMAssay Description:Affinity for rat dopamine transporter using [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50453909(CHEMBL3084880)
Affinity DataKi:  79nMAssay Description:Binding affinity to dopamine transporter (DAT) using [3H]WIN-35428 as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50453909(CHEMBL3084880)
Affinity DataIC50:  468nMAssay Description:Inhibition of [3H]dopamine uptake in rat caudate putamen.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed