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Found 4 Enz. Inhib. hit(s) with Target = 'Sodium-dependent serotonin transporter' and Ligand = 'BDBM50021895'
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM50021895(4-(3,4-Dichloro-phenyl)-7-methoxy-2-methyl-1,2,3,4...)
Affinity DataKi:  3.70nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM50021895(4-(3,4-Dichloro-phenyl)-7-methoxy-2-methyl-1,2,3,4...)
Affinity DataKi:  10nMAssay Description:Inhibition the uptake of tritiated serotonin (5-HT) by the serotonin transporter SERT in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM50021895(4-(3,4-Dichloro-phenyl)-7-methoxy-2-methyl-1,2,3,4...)
Affinity DataKi:  18nMAssay Description:Inhibition of serotonin (5-HT) uptake into rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM50021895(4-(3,4-Dichloro-phenyl)-7-methoxy-2-methyl-1,2,3,4...)
Affinity DataKi:  51nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed