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Found 3 Enz. Inhib. hit(s) with Target = 'Sodium-dependent serotonin transporter' and Ligand = 'BDBM50131357'
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM50131357(4-(5-Fluoro-indan-2-ylmethyl)-4,5-dihydro-1H-imida...)
Affinity DataKi:  25nMAssay Description:In vitro binding affinity was determined against serotonin reuptake site of rat in presence of [3H]paroxetine radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM50131357(4-(5-Fluoro-indan-2-ylmethyl)-4,5-dihydro-1H-imida...)
Affinity DataKi:  77nMAssay Description:In vitro binding affinity towards rat serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50131357(4-(5-Fluoro-indan-2-ylmethyl)-4,5-dihydro-1H-imida...)
Affinity DataKi:  77nMAssay Description:Inhibition of [3H]- paroxetine binding to 5-HTT receptor, serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed