Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Soluble acetylcholine receptor' and Ligand = 'BDBM91615'
TargetSoluble acetylcholine receptor(Aplysia Californica)
University of California San Diego

LigandPNGBDBM91615(15q | alpha7 agonists 15q)
Affinity DataKi:  8nM ΔG°:  -45.4kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSoluble acetylcholine receptor(Aplysia Californica)
University of California San Diego

LigandPNGBDBM91615(15q | alpha7 agonists 15q)
Affinity DataKi:  13nM ΔG°:  -44.3kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSoluble acetylcholine receptor(Aplysia Californica)
University of California San Diego

LigandPNGBDBM91615(15q | alpha7 agonists 15q)
Affinity DataKi:  13nM ΔG°:  -44.3kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed