Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Soluble acetylcholine receptor' and Ligand = 'BDBM91621'
TargetSoluble acetylcholine receptor(Aplysia Californica)
University of California San Diego

LigandPNGBDBM91621(21q | alpha7 agonists 21q)
Affinity DataKi:  18nM ΔG°:  -43.5kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSoluble acetylcholine receptor(Aplysia Californica)
University of California San Diego

LigandPNGBDBM91621(21q | alpha7 agonists 21q)
Affinity DataKi:  30nM ΔG°:  -42.2kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSoluble acetylcholine receptor(Aplysia Californica)
University of California San Diego

LigandPNGBDBM91621(21q | alpha7 agonists 21q)
Affinity DataKi:  400nM ΔG°:  -35.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed