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Found 8 Enz. Inhib. hit(s) with Target = 'Solute carrier family 13 member 5' and Ligand = 'BDBM50149244'
TargetSolute carrier family 13 member 5(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149244(CHEMBL3771118)
Affinity DataIC50:  120nMAssay Description:Inhibition of NaCT in rat hepatocytes assessed as [14C]-citrate uptake after 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149244(CHEMBL3771118)
Affinity DataIC50:  126nMAssay Description:Inhibition of NaCT in rat hepatocytes assessed as [14C]-citrate uptake after 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Mus musculus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149244(CHEMBL3771118)
Affinity DataIC50:  210nMAssay Description:Inhibition of NaCT in mouse hepatocytes assessed as [14C]-citrate uptake after 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Mus musculus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149244(CHEMBL3771118)
Affinity DataIC50:  214nMAssay Description:Inhibition of NaCT in mouse hepatocytes assessed as [14C]-citrate uptake after 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149244(CHEMBL3771118)
Affinity DataIC50:  501nMAssay Description:Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149244(CHEMBL3771118)
Affinity DataIC50:  510nMAssay Description:Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149244(CHEMBL3771118)
Affinity DataIC50:  740nMAssay Description:Inhibition of NaCT in human hepatocytes assessed as [14C]-citrate uptake after 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149244(CHEMBL3771118)
Affinity DataIC50:  794nMAssay Description:Inhibition of NaCT in human hepatocytes assessed as [14C]-citrate uptake after 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed