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Found 2 Enz. Inhib. hit(s) with Target = 'Sortase family protein' and Ligand = 'BDBM50542870'
TargetSortase family protein(Staphylococcus aureus)
Guizhou University

Curated by ChEMBL
LigandPNGBDBM50542870(CHEMBL4637978)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of Staphylococcus aureus SrtA delta N24 mutant expressed in Escherichia coli BL21 (DE3) using Abz-LPATG-Dnp substrate incubated for 20 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSortase family protein(Staphylococcus aureus)
Guizhou University

Curated by ChEMBL
LigandPNGBDBM50542870(CHEMBL4637978)
Affinity DataIC50:  1.67E+4nMAssay Description:Inhibition of Staphylococcus aureus SrtA delta N24 mutant expressed in Escherichia coli BL21 (DE3) assessed as reduction in IsdA (64 to 323 residues)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed