Found 2 Enz. Inhib. hit(s) with Target = 'Sphingosine 1-phosphate receptor 1' and Ligand = 'BDBM50424953' TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Praecis Pharmaceuticals Incorporated (Currently Glaxosmithkline)
Curated by ChEMBL
Praecis Pharmaceuticals Incorporated (Currently Glaxosmithkline)
Curated by ChEMBL
Affinity DataIC50: 95nMAssay Description:Displacement of [33P]S1P from human S1P1 receptor expressed in HEK293T cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Praecis Pharmaceuticals Incorporated (Currently Glaxosmithkline)
Curated by ChEMBL
Praecis Pharmaceuticals Incorporated (Currently Glaxosmithkline)
Curated by ChEMBL
Affinity DataEC50: 135nMAssay Description:Agonist activity at human S1P1 receptor expressed in HEK293T cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
