Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Steryl-sulfatase' and Ligand = 'BDBM24306'
TargetSteryl-sulfatase(Homo sapiens (Human))
University of Bath

LigandPNGBDBM24306(Letrozole derivative, 40 | {2-bromo-4-[(4-cyanophe...)
Affinity DataIC50:  2.60E+3nMAssay Description:The extent of in vitro inhibition of sulfatase activities was assessed using intact monolayers of JEG-3 cells. Sulfatase activity was measured using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University of Bath

LigandPNGBDBM24306(Letrozole derivative, 40 | {2-bromo-4-[(4-cyanophe...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of steroid sulfatase in human JEG-3 cells using [6,7-3H]E1S as substrate after 1 hr by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University of Bath

LigandPNGBDBM24306(Letrozole derivative, 40 | {2-bromo-4-[(4-cyanophe...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of STS activity (unknown origin) expressed in JEG-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed