Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Steryl-sulfatase' and Ligand = 'BDBM50168219'
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50168219(CHEMBL3805209)
Affinity DataIC50:  0.0240nMAssay Description:Inhibition of estrone sulfatase (unknown origin) transfected in HEK293 cells using E1S as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50168219(CHEMBL3805209)
Affinity DataIC50:  0.0500nMAssay Description:Inhibition of steroid sulfatase (unknown origin) expressed in HEK293 cells assessed as reduction in transformation of [3H]-E1S to E1 after 2 hrs by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed