Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Stromelysin-1' and Ligand = 'BDBM8466'
TargetStromelysin-1(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM8466((2R)-N-hydroxy-2-[(4-methoxybenzene)sulfonamido]-3...)
Affinity DataKd:  43nMAssay Description:Binding affinity to stromelysin-1 catalytic domain expressed in Escherichia coli BL21 (DE3) by isothermal titration colorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM8466((2R)-N-hydroxy-2-[(4-methoxybenzene)sulfonamido]-3...)
Affinity DataKd:  113nMAssay Description:Binding affinity to stromelysin-1 catalytic domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed