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Found
1
Enz. Inhib. hit(s) with Target = 'TGF-beta receptor type-1' and Ligand = 'BDBM282795'
Target
TGF-beta receptor type-1
(Homo sapiens (Human))
Rigel Pharmaceuticals
US Patent
Ligand
BDBM282795
(6-(4-(4-fluorophenyl)-1-(3,3,3-trifluoropropyl)-1H...)
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Affinity Data
IC50: 6.80nM
pH: 7.4 T: 2°C
Assay Description:
Assays for the compounds reported below were conducted in 1536-well plates and 2 mL reactions are prepared from addition of HIS-TGF-βR1 T204D or...
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Target Info
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Ligand Info
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US Patent
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