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Found
1
Enz. Inhib. hit(s) with Target = 'TGF-beta receptor type-1' and Ligand = 'BDBM50311017'
Target
TGF-beta receptor type-1
(Homo sapiens (Human))
Gilead Sciences
US Patent
Ligand
BDBM50311017
(CHEMBL1078178 | Momelotinib | N-(cyanomethyl)-4-(2...)
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Affinity Data
IC50: 205nM Kd: 670nM
Assay Description:
Biochemical binding assays (DiscoveRx) and in vitro enzyme inhibition assays (LanthaScreen, Life Technologies) were conducted to determine the bindin...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
antibodypedia
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Ligand Info
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CHEMBL
MCE
PC cid
PC sid
PDB
Patents
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Details
US Patent
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