Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with Target = 'TYR_PHOSPHATASE_2 domain-containing protein' and Ligand = 'BDBM50464771'
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
Universidade Federal De Santa Catarina

Curated by ChEMBL
LigandPNGBDBM50464771(CHEMBL4279417)
Affinity DataKi:  390nMAssay Description:Inhibition of Mycobacterium tuberculosis PtpB using p-nitrophenyl phosphate as substrate preincubated for 10 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
Universidade Federal De Santa Catarina

Curated by ChEMBL
LigandPNGBDBM50464771(CHEMBL4279417)
Affinity DataIC50:  830nMAssay Description:Inhibition of Mycobacterium tuberculosis PtpB using p-nitrophenyl phosphate as substrate preincubated for 10 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
Universidade Federal De Santa Catarina

Curated by ChEMBL
LigandPNGBDBM50464771(CHEMBL4279417)
Affinity DataIC50:  832nMAssay Description:Inhibition of Mycobacterium tuberculosis PtpB using p-nitrophenyl phosphate as substrate preincubated for 10 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
Universidade Federal De Santa Catarina

Curated by ChEMBL
LigandPNGBDBM50464771(CHEMBL4279417)
Affinity DataKd:  700nMAssay Description:Binding affinity to Mycobacterium tuberculosis PtpB by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
Universidade Federal De Santa Catarina

Curated by ChEMBL
LigandPNGBDBM50464771(CHEMBL4279417)
Affinity DataKd:  2.90E+3nMAssay Description:Binding affinity to Mycobacterium tuberculosis PtpB by ITC methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
Universidade Federal De Santa Catarina

Curated by ChEMBL
LigandPNGBDBM50464771(CHEMBL4279417)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity to Mycobacterium tuberculosis PtpB by UV-VIS spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed