Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Trace amine-associated receptor 1' and Ligand = 'BDBM50212653'
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212653(2-(4-phenoxyphenyl)but-3-yn-1-amine hydrochloride ...)
Affinity DataEC50:  929nMAssay Description:Activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212653(2-(4-phenoxyphenyl)but-3-yn-1-amine hydrochloride ...)
Affinity DataEC50:  62nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed